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Drug Name | Lonafarnib |
Trade Name | Sarasar |
Synonyms | SCH66336 |
Drug Descriptions |
Lonafarnib (SCH66336) is a farnesyl transferase inhibitor, which alters post-translational modification and activation of Ras proteins (PMID: 25323927, PMID: 29285232). |
DrugClasses | Farnesyltransferase Inhibitor 3 |
CAS Registry Number | 193275-84-2 |
NCIT ID | C1829 |
Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
---|---|---|---|
Docetaxel + Lonafarnib | Docetaxel Lonafarnib | 0 | 0 |
Lonafarnib | Lonafarnib | 0 | 0 |
Lonafarnib + Tamoxifen | Lonafarnib Tamoxifen | 0 | 0 |