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Drug Name SAR260301
Trade Name
Synonyms SAR 260301|SAR-260301
Drug Descriptions

SAR260301 is PI3K beta-selective inhibitor, which has been demonstrated to inhibit tumor growth in xenograft models (PMID: 24387221, PMID: 28976556).

DrugClasses PIK3CB inhibitor 8
CAS Registry Number 1260612-13-2
NCIT ID C116882

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Therapy Name Drugs Efficacy Evidence Clinical Trials
SAR260301 SAR260301 4 1
SAR260301 + Selumetinib SAR260301 Selumetinib 1 0
SAR260301 + Vemurafenib SAR260301 Vemurafenib 1 1


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