Missing content? – Request curation!
Request curation for specific Genes, Variants, or PubMed publications.
Have questions, comments, or suggestions? - Let us know!
Email us at : ckbsupport@jax.org
Drug Name | Ro 31-8220 |
Trade Name | |
Synonyms | Ro-31-8220|Ro 318220 |
Drug Descriptions |
Ro 31-8220 is a pan-protein kinase C (PKC) inhibitor, with additional activity against additional kinases including GSK3-beta, which may increase apoptosis and decrease growth of tumor cells (PMID: 8373348, PMID: 10998351, PMID: 18281471, PMID: 26657401). |
DrugClasses | GSK-3beta Inhibitor 4 PKC Inhibitor (Pan) 11 |
CAS Registry Number | 125314-64-9 |
NCIT ID | C1310 |
Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
---|---|---|---|
Ro 31-8220 | Ro 31-8220 | 0 | 0 |