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Drug Name E7016
Trade Name
Synonyms E-7016
Drug Descriptions

E7016 is an inhibitor of PARP1 and PARP2, which results in the accumulation of DNA damage, thereby potentially resulting in increased tumor cell death and increased sensitivity to DNA damaging agents (Mol Cancer Ther 2011;10(11 Suppl):Abstract nr B185, PMID: 19147766).

DrugClasses PARP Inhibitor (Pan) 30
CAS Registry Number 902128-92-1
NCIT ID C91387

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Therapy Name Drugs Efficacy Evidence Clinical Trials
E7016 E7016 0 0
E7016 + Temozolomide E7016 Temozolomide 0 0


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