Drug Detail


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Drug Name GSK3052230
Trade Name
Synonyms FP-1039|HGS1036|GSK-3052230|GSK 3052230
Drug Descriptions

GSK3052230 (FP-1039) is an FGF ligand trap which prevents FGF1, FGF2, and FGF4 from binding corresponding receptors thereby preventing downstream signaling and activation (PMID: 26078430, PMID: 31065954, PMID: 31446228).

CAS Registry Number 1631072-93-9
NCIT ID C77970


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Therapy Name Drugs Efficacy Evidence Clinical Trials
Carboplatin + GSK3052230 + Paclitaxel Carboplatin GSK3052230 Paclitaxel 1 0
Cisplatin + Etoposide + GSK3052230 Cisplatin Etoposide GSK3052230 1 0
Cisplatin + GSK3052230 + Pemetrexed Disodium Cisplatin GSK3052230 Pemetrexed Disodium 0 0
GSK3052230 GSK3052230 4 1

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