Drug Detail


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Drug Name Conteltinib
Trade Name
Synonyms CT-707|CT 707
Drug Descriptions

Conteltinib (CT-707) is a kinase inhibitor of FAK (PTK2), PYK2 (PTK2B), ALK, and YAP1 (PMID: 29669759), which may result in antitumor activity including inhibition of both tumor growth and metastasis (PMID: 27638856, PMID: 30381078).

DrugClasses ALK Inhibitor 32 FAK inhibitor 15 YAP Inhibitor 3
CAS Registry Number 1384860-29-0
NCIT ID C126648


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Therapy Name Drugs Efficacy Evidence Clinical Trials
Cabozantinib + Conteltinib Cabozantinib Conteltinib 0 0
Conteltinib Conteltinib 8 0
Conteltinib + PHA-665752 Conteltinib PHA-665752 0 0

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