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Drug Name NPS-1034
Trade Name
Drug Descriptions

NPS-1034 inhibits AXL and MET, including mutant forms of MET, as well as other kinases, which potentially results in decreased tumor cell growth and may overcome MET or AXL mediated drug resistance (PMID: 24173966, PMID: 24165158).

DrugClasses AXL Inhibitor 29 MET Inhibitor 53
CAS Registry Number 1221713-92-3


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Therapy Name Drugs Efficacy Evidence Clinical Trials
Erlotinib + NPS-1034 Erlotinib NPS-1034 0 0
Gefitinib + NPS-1034 Gefitinib NPS-1034 0 0
NPS-1034 NPS-1034 1 0

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