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Drug Name PLX51107
Trade Name
Synonyms PLX-51107|PLX 51107
Drug Descriptions

PLX51107 is a small molecule BET inhibitor, which binds to BET bromodomains in BRD2, BRD3, BRD4, and BRDT, potentially resulting in decreased tumor cell proliferation (PMID: 29386193, PMID: 31063649, PMID: 32717030).

DrugClasses BET Inhibitor (Pan) 32
CAS Registry Number 1627929-55-8
NCIT ID C125739

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Therapy Name Drugs Efficacy Evidence Clinical Trials
Azacitidine + PLX51107 Azacitidine PLX51107 0 1
PLX51107 PLX51107 0 1


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