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Drug Name | RAD140 |
Trade Name | |
Synonyms | RAD-140|RAD 140 |
Drug Descriptions |
RAD140, a selective androgen receptor modulator, results in AR agonist activity, thereby regulating AR target genes and repressing ESR1, which may inhibit the growth of tumors expressing AR and ESR1 (PMID: 28974548). |
DrugClasses | Hormone - Anti-androgens 38 |
CAS Registry Number | 1182367-47-0 |
NCIT ID | C137950 |
Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
---|---|---|---|
Palbociclib + RAD140 | Palbociclib RAD140 | 0 | 0 |
RAD140 | RAD140 | 0 | 1 |