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Drug Name RAD140
Trade Name
Synonyms RAD-140|RAD 140
Drug Descriptions

RAD140, a selective androgen receptor modulator, results in AR agonist activity, thereby regulating AR target genes and repressing ESR1, which may inhibit the growth of tumors expressing AR and ESR1 (PMID: 28974548).

DrugClasses Hormone - Anti-androgens 38
CAS Registry Number 1182367-47-0
NCIT ID C137950


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Therapy Name Drugs Efficacy Evidence Clinical Trials
Palbociclib + RAD140 Palbociclib RAD140 0 0
RAD140 RAD140 0 1

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