Drug Detail


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Drug Name BGB3245
Trade Name
Synonyms BGB-3245|BGB 3245
Drug Descriptions

BGB3245 inhibits RAF dimer formation, which may lead to inhibition of Erk signaling and cell growth (PMID: 29880583).

DrugClasses RAF Inhibitor (Pan) 27
CAS Registry Number NA
NCIT ID C173633


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Therapy Name Drugs Efficacy Evidence Clinical Trials
BGB3245 BGB3245 6 1
BGB3245 + Panitumumab BGB3245 Panitumumab 0 1
BGB3245 + PD-0325901 BGB3245 PD-0325901 0 1

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