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Drug Name UNC0642
Trade Name
Synonyms MP-IN-317
Drug Descriptions

UNC0642 (MP-IN-317) is a histone methyltransferase inhibitor that selectively inhibits EHMT2 (G9A) and EHMT1 (GLP), which may result in decreased methylation and potential cytotoxic effects against cancer cells (PMID: 24102134).

DrugClasses EHMT2 Inhibitor 5
CAS Registry Number NA
NCIT ID NA

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Therapy Name Drugs Efficacy Evidence Clinical Trials
Afatinib + UNC0642 Afatinib UNC0642 0 0
UNC0642 UNC0642 0 0


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