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Drug Name Megestrol acetate
Trade Name Megace
Synonyms MGA|Linmegestrol|Magestin|Megestat|Megeron
Drug Descriptions

Megace (megestrol acetate) is a progestin that activates progesterone receptor signaling and blocks luteinizing hormone signaling, which may lead to potential anti-estrogen and antitumor activities (PMID: 2471590).

CAS Registry Number 3562-63-8


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Therapy Name Drugs Efficacy Evidence Clinical Trials
Ipatasertib + Megestrol acetate Ipatasertib Megestrol acetate 0 1
Letrozole + Megestrol acetate Letrozole Megestrol acetate 0 1
Megestrol acetate Megestrol acetate 0 5
Megestrol acetate + Pterostilbene Megestrol acetate Pterostilbene 0 1
Megestrol acetate + Sodium cridanimod Megestrol acetate Sodium cridanimod 0 1

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