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Drug Name BI2536
Trade Name
Synonyms BI 2536|BI-2536
Drug Descriptions

BI2536 inhibits polo-like kinase 1 (PLK1), which disrupts mitosis and induces apoptosis in tumor cells (PMID: 30414309, PMID: 32486290).

DrugClasses PLK1 Inhibitor 17
CAS Registry Number 755038-02-9
NCIT ID C49091

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Therapy Name Drugs Efficacy Evidence Clinical Trials
BI2536 BI2536 1 0
BI2536 + Metformin BI2536 Metformin 0 0
BI2536 + PD-0325901 BI2536 PD-0325901 0 0
BI2536 + PLX4720 BI2536 PLX4720 1 0


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