Drug Detail


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Drug Name E6201
Trade Name
Drug Descriptions

E6201 is a dual inhibitor of MEK1 and FLT3, which may lead to decreased tumor cell growth (Blood Nov 2013, 122 (21) 2683; PMID: 23039341, PMID: 29867224, PMID: 30264293).

DrugClasses FLT3 Inhibitor 66 MEK1 Inhibitor 26
CAS Registry Number 603987-35-5
NCIT ID C79848


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Therapy Name Drugs Efficacy Evidence Clinical Trials
Dabrafenib + E6201 Dabrafenib E6201 0 2
E6201 E6201 20 2
E6201 + E7449 E6201 E7449 0 0
E6201 + LY294002 E6201 LY294002 1 0

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