Drug Detail


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Drug Name LY294002
Trade Name
Synonyms LY-294002|LY 294002|NSC-697286|SF-1101
Drug Descriptions

LY294002 is a specific inhibitor of PI3K alpha, beta, and delta, which leads to inhibition of PI3K-Akt/PKB signaling (PMID: 12060641, PMID: 31759362, PMID: 31732769).

DrugClasses PI3K Inhibitor (Pan) 40
CAS Registry Number 154447-36-6
NCIT ID C148229


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Therapy Name Drugs Efficacy Evidence Clinical Trials
Cisplatin + LY294002 Cisplatin LY294002 1 0
E6201 + LY294002 E6201 LY294002 1 0
Gefitinib + LY294002 Gefitinib LY294002 0 0
Imatinib + LY294002 Imatinib LY294002 1 0
LY294002 LY294002 1 0
LY294002 + RU-SKI 43 LY294002 RU-SKI 43 0 0
LY294002 + Sirolimus LY294002 Sirolimus 0 0

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