Drug Detail


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Drug Name GSK2256098
Trade Name
Synonyms GSK-2256098|GSK 2256098
Drug Descriptions

GSK2256098 is an inhibitor of focal adhesion kinase (FAK), which blocks integrin signaling and therefore, has antitumor activities (PMID: 21787277, PMID: 30992546).

DrugClasses FAK inhibitor 15
CAS Registry Number 1224887-10-8
NCIT ID C88346


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Therapy Name Drugs Efficacy Evidence Clinical Trials
Cisplatin + GSK2256098 Cisplatin GSK2256098 0 0
GSK2256098 GSK2256098 2 1
GSK2256098 + Paclitaxel GSK2256098 Paclitaxel 1 0
GSK2256098 + Topotecan GSK2256098 Topotecan 1 0
GSK2256098 + Trametinib GSK2256098 Trametinib 0 1

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