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Drug Name AR-42
Trade Name
Synonyms HDAC42
Drug Descriptions

AR-42 is a histone deacetylase (HDAC) inhibitor, which may lead to increased apoptosis of tumor cells and decreased tumor growth (PMID: 23178755, PMID: 21778190).

DrugClasses HDAC Inhibitor 38
CAS Registry Number 935881-37-1
NCIT ID C116850


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Therapy Name Drugs Efficacy Evidence Clinical Trials
AR-42 AR-42 4 1
AR-42 + Cisplatin AR-42 Cisplatin 1 0
AR-42 + Decitabine AR-42 Decitabine 1 1
AR-42 + Dexamethasone + Pomalidomide AR-42 Dexamethasone Pomalidomide 0 1
AR-42 + Pazopanib AR-42 Pazopanib 0 1

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