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Drug Name Pazopanib
Trade Name Votrient
Synonyms GW-786034
Drug Descriptions

Votrient (pazopanib) inhibits VEGFR-1, -2 and -3, KIT, and PDGFR, and FGFR1, 2, and 3, leading to decreased tumor angiogenesis and growth (PMID: 17620431, PMID: 23786770). Votrient (pazopanib) is approved for renal cell carcinoma and soft tissue sarcoma (FDA.gov).

DrugClasses FGFR1 Inhibitor 28 FGFR2 Inhibitor 23 FGFR3 Inhibitor 19 KIT Inhibitor 57 PDGFR Inhibitor (Pan) 30 VEGFR Inhibitor (Pan) 36
CAS Registry Number 444731-52-6
NCIT ID C74547

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Therapy Name Drugs Efficacy Evidence Clinical Trials
Abexinostat + Pazopanib Abexinostat Pazopanib 0 1
Alisertib + Pazopanib Alisertib Pazopanib 0 1
Bevacizumab + Pazopanib Bevacizumab Pazopanib 0 1
Carboplatin + Paclitaxel + Pazopanib Carboplatin Paclitaxel Pazopanib 0 0
Carotuximab + Pazopanib Carotuximab Pazopanib 0 3
Cetuximab + Pazopanib Cetuximab Pazopanib 0 1
Crizotinib + Pazopanib Crizotinib Pazopanib 2 1
Crizotinib + Pazopanib + Pemetrexed Disodium Crizotinib Pazopanib Pemetrexed Disodium 0 1
Dabrafenib + Pazopanib Dabrafenib Pazopanib 0 1
Docetaxel + Gemcitabine + Pazopanib Docetaxel Gemcitabine Pazopanib 0 2
Docetaxel + Pazopanib + Pegfilgrastim Docetaxel Pazopanib Pegfilgrastim 0 1
Doxorubicin + Ifosfamide + Pazopanib Doxorubicin Ifosfamide Pazopanib 0 1
Everolimus + Pazopanib Everolimus Pazopanib 0 1
Evofosfamide + Pazopanib Evofosfamide Pazopanib 0 1
Gemcitabine + Pazopanib Gemcitabine Pazopanib 0 4
Irinotecan + Pazopanib + Temozolomide Irinotecan Pazopanib Temozolomide 0 1
Nab-rapamycin + Pazopanib Nab-rapamycin Pazopanib 0 1
Nivolumab + Pazopanib Nivolumab Pazopanib 0 1
Paclitaxel + Pazopanib Paclitaxel Pazopanib 0 3
Panobinostat + Pazopanib Panobinostat Pazopanib 0 1
Pazopanib Pazopanib 15 50
Pazopanib + Pembrolizumab Pazopanib Pembrolizumab 0 0
Pazopanib + Pemetrexed Disodium Pazopanib Pemetrexed Disodium 0 1
Pazopanib + PRT1419 PRT1419 Pazopanib 0 0
Pazopanib + REC-2282 Pazopanib REC-2282 0 1
Pazopanib + Siremadlin Pazopanib Siremadlin 0 1
Pazopanib + Spartalizumab Pazopanib Spartalizumab 0 1
Pazopanib + Sunitinib Pazopanib Sunitinib 0 1
Pazopanib + Temozolomide Pazopanib Temozolomide 0 1
Pazopanib + Topotecan Pazopanib Topotecan 0 5
Pazopanib + Trabectedin Pazopanib Trabectedin 0 0
Pazopanib + Trametinib Pazopanib Trametinib 1 1
Pazopanib + Trebananib Pazopanib Trebananib 0 1
Pazopanib + Vorinostat Pazopanib Vorinostat 4 0


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