Drug Detail

Contact

Missing content? – Request curation!

Request curation for specific Genes, Variants, or PubMed publications.

Have questions, comments, or suggestions? - Let us know!

Email us at : ckbsupport@jax.org

Drug Name Alisertib
Trade Name
Synonyms MLN8237
Drug Descriptions

Alisertib (MLN8237) binds to and inhibits Aurora A kinase, which may result in disruption of the assembly of the mitotic spindle apparatus, disruption of chromosome segregation, and inhibition of cell proliferation (PMID: 26999067, PMID: 32414750).

DrugClasses Aurka Inhibitors 26
CAS Registry Number 1028486-01-2
NCIT ID C71717

Filtering

  • Case insensitive filtering will display rows if any text in any cell matches the filter term
  • Use simple literal full or partial string matches
  • Separate multiple filter terms with a space. Any order may be used (i. e. a b c and c b a are equivalent )
  • Filtering will only apply to rows that are already loaded on the page. Filtering has no impact on query parameters.
  • Use quotes to match on a longer phrase with spaces (i.e. "mtor c1483f")

Sorting

  • Generally, the default sort order for tables is set to be first column ascending; however, specific tables may set a different default sort order.
  • Click on any column header arrows to sort by that column
  • Hold down the Shift key and click multiple columns to sort by more than one column. Be sure to set ascending or descending order for a given column before moving on to the next column.

Therapy Name Drugs Efficacy Evidence Clinical Trials
Abiraterone + Alisertib + Prednisone Abiraterone Alisertib Prednisone 0 0
Alisertib Alisertib 0 20
Alisertib + Anastrozole Alisertib Anastrozole 0 0
Alisertib + Bortezomib + Rituximab Alisertib Bortezomib Rituximab 0 1
Alisertib + Brentuximab vedotin Alisertib Brentuximab vedotin 0 1
Alisertib + Carboplatin + Cyclophosphamide + Etoposide Alisertib Carboplatin Cyclophosphamide Etoposide 0 1
Alisertib + Carboplatin + Cyclophosphamide + Vincristine Sulfate Alisertib Carboplatin Cyclophosphamide Vincristine Sulfate 0 1
Alisertib + Cetuximab Alisertib Cetuximab 0 1
Alisertib + Cisplatin Alisertib Cisplatin 0 0
Alisertib + Cisplatin + Cyclophosphamide + Vincristine Sulfate Alisertib Cisplatin Cyclophosphamide Vincristine Sulfate 0 1
Alisertib + Cisplatin + Etoposide Alisertib Cisplatin Etoposide 0 0
Alisertib + Docetaxel Alisertib Docetaxel 0 0
Alisertib + Eribulin Alisertib Eribulin 0 0
Alisertib + Esomeprazole Alisertib Esomeprazole 0 1
Alisertib + Etoposide Alisertib Etoposide 0 0
Alisertib + Exemestane Alisertib Exemestane 0 0
Alisertib + Fulvestrant Alisertib Fulvestrant 0 1
Alisertib + Gemcitabine Alisertib Gemcitabine 0 1
Alisertib + Irinotecan Alisertib Irinotecan 0 1
Alisertib + Irinotecan + Temozolomide Alisertib Irinotecan Temozolomide 0 1
Alisertib + Letrozole Alisertib Letrozole 0 0
Alisertib + Mobocertinib Alisertib Mobocertinib 0 0
Alisertib + MP7 Alisertib MP7 0 0
Alisertib + Nab-paclitaxel Alisertib Nab-paclitaxel 0 1
Alisertib + Neratinib Alisertib Neratinib 0 0
Alisertib + Osimertinib Alisertib Osimertinib 0 2
Alisertib + Paclitaxel Alisertib Paclitaxel 0 1
Alisertib + Palbociclib Alisertib Palbociclib 2 0
Alisertib + Pazopanib Alisertib Pazopanib 0 1
Alisertib + Pembrolizumab Alisertib Pembrolizumab 0 1
Alisertib + Rifampin Alisertib Rifampin 0 1
Alisertib + Rituximab Alisertib Rituximab 0 0
Alisertib + Rituximab + Vincristine Sulfate Alisertib Rituximab Vincristine Sulfate 0 0
Alisertib + Sapanisertib Alisertib Sapanisertib 0 2
Alisertib + Tamoxifen Alisertib Tamoxifen 0 0
Alisertib + Tovorafenib Alisertib Tovorafenib 0 1
Alisertib + Vandetanib Alisertib Vandetanib 0 0
Alisertib + Venetoclax Alisertib Venetoclax 0 0
Alisertib + Vorinostat Alisertib Vorinostat 0 0


Additional content available in CKB BOOST