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Drug Name CPI-0610
Trade Name
Synonyms CPI0610
Drug Descriptions

CPI-0610 is a small molecule that binds to BET bromodomains and inhibits interaction with acetylated histones, resulting in regulation of BET-dependent gene expression and anti-tumor effects (PMID: 26815195, PMID: 31729905).

DrugClasses BET Inhibitor (Pan) 32
CAS Registry Number 1380087-89-7
NCIT ID C111901

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Therapy Name Drugs Efficacy Evidence Clinical Trials
CPI-0610 CPI-0610 0 4
CPI-0610 + Dasatinib CPI-0610 Dasatinib 0 0
CPI-0610 + Dasatinib + Rucaparib CPI-0610 Dasatinib Rucaparib 0 0
CPI-0610 + Doxorubicin CPI-0610 Doxorubicin 0 0
CPI-0610 + Rucaparib CPI-0610 Rucaparib 0 0
CPI-0610 + Ruxolitinib CPI-0610 Ruxolitinib 0 2


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