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Drug Name YK-4-279
Trade Name
Drug Descriptions

YK-4-279 is a small molecule inhibitor of the ETS transcription factors, ERG and ETV1, which may result in inhibition of cell mobility and invasion (PMID: 21559405, PMID: 32016454).

CAS Registry Number 1037184-44-3


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Therapy Name Drugs Efficacy Evidence Clinical Trials
Enzastaurin + YK-4-279 Enzastaurin YK-4-279 0 0
Lenalidomide + YK-4-279 Lenalidomide YK-4-279 0 0
TK216 + YK-4-279 TK216 YK-4-279 0 0
Venetoclax + YK-4-279 Venetoclax YK-4-279 0 0
YK-4-279 YK-4-279 0 0

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