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Drug Name TK216
Trade Name
Synonyms TK-216|TK 216
Drug Descriptions

TK216 binds to and inhibits Ets-family transcription factor, which may lead to anti-tumor effects (PMID: 31182435).

CAS Registry Number 1903783-48-1
NCIT ID C125657


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Therapy Name Drugs Efficacy Evidence Clinical Trials
Decitabine + TK216 Decitabine TK216 0 1
Lenalidomide + TK216 Lenalidomide TK216 0 0
Pomalidomide + TK216 Pomalidomide TK216 0 0
TK216 TK216 0 2
TK216 + Venetoclax TK216 Venetoclax 0 0
TK216 + YK-4-279 TK216 YK-4-279 0 0

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