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Drug Name Elraglusib
Trade Name
Synonyms 9 ING 41|9-ING-41
Drug Descriptions

Elraglusib is an ATP-competitive inhibitor that selectively blocks GSK-3beta, potentially leading to cell cycle arrest and apoptosis, inhibition of tumor cell proliferation, and decreased tumor growth (PMID: 31894292, PMID: 29846250).

DrugClasses GSK-3beta Inhibitor 4
CAS Registry Number 1034895-42-5
NCIT ID C156792

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Therapy Name Drugs Efficacy Evidence Clinical Trials
Carboplatin + Elraglusib Carboplatin Elraglusib 0 3
Carboplatin + Elraglusib + Paclitaxel Carboplatin Elraglusib Paclitaxel 0 1
Docetaxel + Elraglusib + Gemcitabine Docetaxel Elraglusib Gemcitabine 0 2
Doxorubicin + Elraglusib Doxorubicin Elraglusib 0 1
Elraglusib Elraglusib 0 2
Elraglusib + Fluorouracil + Irinotecan + Leucovorin + Losartan + Oxaliplatin Elraglusib Fluorouracil Irinotecan Leucovorin Losartan Oxaliplatin 0 1
Elraglusib + Fluorouracil + Irinotecan + Leucovorin + Oxaliplatin Elraglusib Fluorouracil Irinotecan Leucovorin Oxaliplatin 0 1
Elraglusib + Gemcitabine Elraglusib Gemcitabine 0 1
Elraglusib + Gemcitabine + Nab-paclitaxel Elraglusib Gemcitabine Nab-paclitaxel 0 1
Elraglusib + Gemcitabine + Nab-paclitaxel + Retifanlimab Elraglusib Gemcitabine Nab-paclitaxel Retifanlimab 0 1
Elraglusib + Irinotecan Elraglusib Irinotecan 0 2
Elraglusib + Lomustine Elraglusib Lomustine 0 1


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