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Drug Name Tegafur-gimeracil-oteracil Potassium
Trade Name
Synonyms TS-1|BMS-247616
Drug Descriptions

Tegafur-gimeracil-oteracil Potassium (TS-1) is composed of tegafur, gimestat and otastat potassium, of which the ultimate active ingredient is 5-FU (PMID: 12066214, PMID: 32233637).

DrugClasses Chemotherapy - Antimetabolite 14
CAS Registry Number 154239-56-2
NCIT ID C1833

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Therapy Name Drugs Efficacy Evidence Clinical Trials
AZD2936 + Gemcitabine + Tegafur-gimeracil-oteracil Potassium AZD2936 Gemcitabine Tegafur-gimeracil-oteracil Potassium 0 0
AZD2936 + Tegafur-gimeracil-oteracil Potassium AZD2936 Tegafur-gimeracil-oteracil Potassium 0 1
Bemarituzumab + Nivolumab + Oxaliplatin + Tegafur-gimeracil-oteracil Potassium Bemarituzumab Nivolumab Oxaliplatin Tegafur-gimeracil-oteracil Potassium 0 1
Capecitabine + Nivolumab + Oxaliplatin + Tegafur-gimeracil-oteracil Potassium Capecitabine Nivolumab Oxaliplatin Tegafur-gimeracil-oteracil Potassium 0 0
Cisplatin + Durvalumab + Gemcitabine + Tegafur-gimeracil-oteracil Potassium Cisplatin Durvalumab Gemcitabine Tegafur-gimeracil-oteracil Potassium 0 1
Cisplatin + Tegafur-gimeracil-oteracil Potassium Cisplatin Tegafur-gimeracil-oteracil Potassium 0 0
Durvalumab + Gemcitabine + Tegafur-gimeracil-oteracil Potassium Durvalumab Gemcitabine Tegafur-gimeracil-oteracil Potassium 0 1
Nivolumab + Oxaliplatin + RO7496353 + Tegafur-gimeracil-oteracil Potassium Nivolumab Oxaliplatin RO7496353 Tegafur-gimeracil-oteracil Potassium 0 1
Nivolumab + Relatlimab + Tegafur-gimeracil-oteracil Potassium Nivolumab Relatlimab Tegafur-gimeracil-oteracil Potassium 0 1
Nivolumab + Tegafur-gimeracil-oteracil Potassium Nivolumab Tegafur-gimeracil-oteracil Potassium 0 1
Oxaliplatin + Pembrolizumab + Tegafur-gimeracil-oteracil Potassium + Trastuzumab Oxaliplatin Pembrolizumab Tegafur-gimeracil-oteracil Potassium Trastuzumab 0 1
Oxaliplatin + Ramucirumab + Tegafur-gimeracil-oteracil Potassium Oxaliplatin Ramucirumab Tegafur-gimeracil-oteracil Potassium 0 0
Oxaliplatin + Tegafur-gimeracil-oteracil Potassium + Toripalimab-tpzi Oxaliplatin Tegafur-gimeracil-oteracil Potassium Toripalimab-tpzi 0 0
Oxaliplatin + Tegafur-gimeracil-oteracil Potassium + Trastuzumab Oxaliplatin Tegafur-gimeracil-oteracil Potassium Trastuzumab 0 1
Paclitaxel + Tegafur-gimeracil-oteracil Potassium Paclitaxel Tegafur-gimeracil-oteracil Potassium 0 0
Rivoceranib + Tegafur-gimeracil-oteracil Potassium Rivoceranib Tegafur-gimeracil-oteracil Potassium 0 0
TAS-114 + Tegafur-gimeracil-oteracil Potassium TAS-114 Tegafur-gimeracil-oteracil Potassium 0 1
Tegafur-gimeracil-oteracil Potassium Tegafur-gimeracil-oteracil Potassium 0 2
Tegafur-gimeracil-oteracil Potassium + Trastuzumab Tegafur-gimeracil-oteracil Potassium Trastuzumab 0 0


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