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Drug Name Trifluridine-tipiracil hydrochloride
Trade Name Lonsurf
Synonyms TAS-102|TAS102|TAS 102|S 95005|S95005|S-95005
Drug Descriptions

Lonsurf (trifluridine/tipiracil hydrochloride) is an oral combination comprised of TFT and a thymidine phosphorylase inhibitor, which can result in DNA fragmentation thereby preventing angiogenesis and tumor growth and is FDA approved for use in patients with colorectal cancer, gastric or gastroesophageal junction adenocarcinoma (FDA.gov).

DrugClasses
CAS Registry Number 183204-74-2
NCIT ID C102554

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Therapy Name Drugs Efficacy Evidence Clinical Trials
Bevacizumab + Capecitabine + Trifluridine-tipiracil hydrochloride Bevacizumab Capecitabine Trifluridine-tipiracil hydrochloride 0 1
Bevacizumab + Irinotecan + Oxaliplatin + Trifluridine-tipiracil hydrochloride Bevacizumab Irinotecan Oxaliplatin Trifluridine-tipiracil hydrochloride 0 1
Bevacizumab + Irinotecan + Trifluridine-tipiracil hydrochloride Bevacizumab Irinotecan Trifluridine-tipiracil hydrochloride 0 1
Bevacizumab + MM-398 + Trifluridine-tipiracil hydrochloride Bevacizumab MM-398 Trifluridine-tipiracil hydrochloride 0 1
Bevacizumab + Trifluridine-tipiracil hydrochloride Bevacizumab Trifluridine-tipiracil hydrochloride 0 3
CA102N + Trifluridine-tipiracil hydrochloride CA102N Trifluridine-tipiracil hydrochloride 0 1
Cabozantinib + Trifluridine-tipiracil hydrochloride Cabozantinib Trifluridine-tipiracil hydrochloride 0 1
Irinotecan + Trifluridine-tipiracil hydrochloride Irinotecan Trifluridine-tipiracil hydrochloride 0 1
MM-398 + Trifluridine-tipiracil hydrochloride MM-398 Trifluridine-tipiracil hydrochloride 0 1
Nivolumab + Trifluridine-tipiracil hydrochloride Nivolumab Trifluridine-tipiracil hydrochloride 0 1
Panitumumab + Trifluridine-tipiracil hydrochloride Panitumumab Trifluridine-tipiracil hydrochloride 0 1
PolyPEPI1018 + Trifluridine-tipiracil hydrochloride PolyPEPI1018 Trifluridine-tipiracil hydrochloride 0 1
Ramucirumab + Trifluridine-tipiracil hydrochloride Ramucirumab Trifluridine-tipiracil hydrochloride 0 4
Regorafenib + Trifluridine-tipiracil hydrochloride Regorafenib Trifluridine-tipiracil hydrochloride 0 5
Rivoceranib + Trifluridine-tipiracil hydrochloride Rivoceranib Trifluridine-tipiracil hydrochloride 0 1
Talazoparib + Trifluridine-tipiracil hydrochloride Talazoparib Trifluridine-tipiracil hydrochloride 0 1
Trametinib + Trifluridine-tipiracil hydrochloride Trametinib Trifluridine-tipiracil hydrochloride 0 1
Trastuzumab + Trifluridine-tipiracil hydrochloride + Tucatinib Trastuzumab Trifluridine-tipiracil hydrochloride Tucatinib 0 1
Trifluridine-tipiracil hydrochloride Trifluridine-tipiracil hydrochloride 0 16
Trifluridine-tipiracil hydrochloride + UCB6114 Trifluridine-tipiracil hydrochloride UCB6114 0 1


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