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Drug Name Ulixertinib
Trade Name
Synonyms BVD-523|BVD 523|BVD523
Drug Descriptions

Ulixertinib (BVD-523) inhibits both ERK 1 and 2, thereby preventing the activation of ERK-mediated signal transduction pathways and resulting in growth inhibition (PMID: 28939558).

DrugClasses ERK Inhibitor (pan) 21
CAS Registry Number 869886-67-9
NCIT ID C104744

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Therapy Name Drugs Efficacy Evidence Clinical Trials
AZD8186 + Ulixertinib AZD8186 Ulixertinib 0 0
Binimetinib + Ulixertinib Binimetinib Ulixertinib 1 0
Cetuximab + Encorafenib + Ulixertinib Cetuximab Encorafenib Ulixertinib 1 1
Cetuximab + Ulixertinib Cetuximab Ulixertinib 0 1
Gemcitabine + Nab-paclitaxel + Ulixertinib Gemcitabine Nab-paclitaxel Ulixertinib 0 1
Hydroxychloroquine + Ulixertinib Hydroxychloroquine Ulixertinib 0 2
JQ1 + Ulixertinib JQ1 Ulixertinib 1 0
Lifirafenib + Ulixertinib Lifirafenib Ulixertinib 2 0
MRTX-1133 + Ulixertinib MRTX-1133 Ulixertinib 0 0
Navitoclax + Ulixertinib Navitoclax Ulixertinib 1 0
Palbociclib + Ulixertinib Palbociclib Ulixertinib 1 1
Repotrectinib + Ulixertinib Repotrectinib Ulixertinib 0 0
Selpercatinib + Ulixertinib Selpercatinib Ulixertinib 0 0
Selumetinib + Ulixertinib Selumetinib Ulixertinib 1 0
SHP099 + Ulixertinib SHP099 Ulixertinib 1 0
Tipifarnib + Ulixertinib Tipifarnib Ulixertinib 2 0
Trametinib + Ulixertinib Trametinib Ulixertinib 1 0
Ulixertinib Ulixertinib 31 8
Ulixertinib + Vinblastine Ulixertinib Vinblastine 1 0


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