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| Drug Name | SHP099 |
| Trade Name | |
| Synonyms | SHP-099|SHP 099 |
| Drug Descriptions |
SHP099 is an allosteric inhibitor of SHP2 that stabilizes SHP2 in its autoinhibited conformation, which reduces downstream signaling and potentially leads to decreased growth of receptor tyrosine kinase-driven tumors (PMID: 27362227, PMID: 31043123). |
| DrugClasses | SHP2 Inhibitor 19 |
| CAS Registry Number | 1801747-42-4 |
| NCIT ID | NA |
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