Drug Detail

Contact

Missing content? – Request curation!

Request curation for specific Genes, Variants, or PubMed publications.

Have questions, comments, or suggestions? - Let us know!

Email us at : ckbsupport@jax.org

Drug Name Epacadostat
Trade Name
Synonyms INCB024360|INCB 024360|INCB-024360
Drug Descriptions

Epacadostat (INCB024360) inhibits indoleamine 2,3-dioxygenase 1 (IDO1) to prevent conversion of tryptophan to kynurenine, potentially resulting in increased proliferation of T-cells and natural killer cells and enhanced anti-tumor immune response (PMID: 20197554).

DrugClasses IDO1 Inhibitor 12
CAS Registry Number 1204669-58-8
NCIT ID C92582

Filtering

  • Case insensitive filtering will display rows if any text in any cell matches the filter term
  • Use simple literal full or partial string matches
  • Separate multiple filter terms with a space. Any order may be used (i. e. a b c and c b a are equivalent )
  • Filtering will only apply to rows that are already loaded on the page. Filtering has no impact on query parameters.
  • Use quotes to match on a longer phrase with spaces (i.e. "mtor c1483f")

Sorting

  • Generally, the default sort order for tables is set to be first column ascending; however, specific tables may set a different default sort order.
  • Click on any column header arrows to sort by that column
  • Hold down the Shift key and click multiple columns to sort by more than one column. Be sure to set ascending or descending order for a given column before moving on to the next column.

Therapy Name Drugs Efficacy Evidence Clinical Trials
ALT-803 + Bintrafusp alfa + Epacadostat + FPV-Brachyury + MVA-BN-Brachyury ALT-803 Bintrafusp alfa Epacadostat FPV-Brachyury MVA-BN-Brachyury 0 1
Atezolizumab + Epacadostat Atezolizumab Epacadostat 0 1
Avelumab + Bevacizumab + Epacadostat Avelumab Bevacizumab Epacadostat 0 0
Azacitidine + Epacadostat + Pembrolizumab Azacitidine Epacadostat Pembrolizumab 0 1
Bevacizumab + Epacadostat + Radiotherapy + Retifanlimab Bevacizumab Epacadostat Radiotherapy Retifanlimab 0 1
Carboplatin + Cisplatin + Epacadostat + Fluorouracil + Nivolumab Carboplatin Cisplatin Epacadostat Fluorouracil Nivolumab 0 1
Carboplatin + Cisplatin + Epacadostat + Gemcitabine + Nivolumab + Paclitaxel + Pemetrexed Disodium Carboplatin Cisplatin Epacadostat Gemcitabine Nivolumab Paclitaxel Pemetrexed Disodium 0 1
Carboplatin + Epacadostat + Paclitaxel + Pembrolizumab Carboplatin Epacadostat Paclitaxel Pembrolizumab 0 2
Carboplatin + Epacadostat + Pembrolizumab + Pemetrexed Disodium Carboplatin Epacadostat Pembrolizumab Pemetrexed Disodium 0 2
Cisplatin + Epacadostat + Pembrolizumab + Pemetrexed Disodium Cisplatin Epacadostat Pembrolizumab Pemetrexed Disodium 0 1
CRS-207 + Cyclophosphamide + Epacadostat + GVAX pancreatic cancer vaccine + Pembrolizumab CRS-207 Cyclophosphamide Epacadostat GVAX pancreatic cancer vaccine Pembrolizumab 0 1
CRS-207 + Epacadostat + Pembrolizumab CRS-207 Epacadostat Pembrolizumab 0 1
Cyclophosphamide + Epacadostat + Maveropepimut-S Cyclophosphamide Epacadostat Maveropepimut-S 0 1
Cyclophosphamide + Epacadostat + Pembrolizumab Cyclophosphamide Epacadostat Pembrolizumab 0 1
Durvalumab + Epacadostat Durvalumab Epacadostat 0 2
Epacadostat Epacadostat 0 8
Epacadostat + Fluorouracil + Leucovorin + Nivolumab + Oxaliplatin Epacadostat Fluorouracil Leucovorin Nivolumab Oxaliplatin 0 1
Epacadostat + Gemcitabine + Nab-paclitaxel + Nivolumab Epacadostat Gemcitabine Nab-paclitaxel Nivolumab 0 1
Epacadostat + INCAGN01876 + Pembrolizumab Epacadostat INCAGN01876 Pembrolizumab 0 1
Epacadostat + INCB001158 Epacadostat INCB001158 0 1
Epacadostat + INCB001158 + Pembrolizumab Epacadostat INCB001158 Pembrolizumab 0 1
Epacadostat + Ipilimumab + Nivolumab Epacadostat Ipilimumab Nivolumab 0 1
Epacadostat + Itacitinib Epacadostat Itacitinib 0 1
Epacadostat + Lirilumab + Nivolumab Epacadostat Lirilumab Nivolumab 0 1
Epacadostat + Nivolumab Epacadostat Nivolumab 0 2
Epacadostat + OATD-02 + unspecified PD-L1 antibody Epacadostat OATD-02 unspecified PD-L1 antibody 0 0
Epacadostat + Pembrolizumab Epacadostat Pembrolizumab 0 20
Epacadostat + Pembrolizumab + Tavokinogene telseplasmid Epacadostat Pembrolizumab Tavokinogene telseplasmid 0 1
Epacadostat + Retifanlimab Epacadostat Retifanlimab 0 3
Epacadostat + SD-101 Epacadostat SD-101 0 1
Epacadostat + Sirolimus Epacadostat Sirolimus 0 1


Additional content available in CKB BOOST